Anastrozole (Arimidex) is a selective and competitive nonsteroidal aromatase inhibitor of a new generation. The effect of drugs in this group is to reduce the level of estrogen in the blood by completely inhibiting the peripheral action of aromatase, without affecting other hormones. The active ingredient of the drug is anastrozole.
At 1 mg and 10 mg, it inhibits the aromatization of androstenedione in 96.7%. and 98.1%, while estrone and estradiol levels decreased by 86.5% and 83.5%. Knowledge of the clinical properties of Arimidex and its possible uses increase with the results of subsequent trials. It can be said that it is more effective than tamoxifen. In bodybuilding, it is used when taking drugs that are highly aromatic and vulnerable to gynecomastia. Anastrozole has a minimal amount of side effects and can severely block the formation of estrogen. He works on the cause of estrogen formation, and not as new, Proviron or Clomid, which only block estrogen receptors.
Anastrozole - is an oral aromatase inhibitor manufactured by Zeneca Pharmaceuticals and approved for use in the United States in 1995. This drug is licensed, so you need a written doctor's prescription to get it. It is primarily prescribed for the adjutant therapy of postmenopausal women with breast cancer with hormone receptors. Adjutant therapy - is a treatment given in addition to the primary treatment of a patient to prevent the multiplication of cancer cells.
Anastrozole - was the first selective aromatase inhibitor used in bodybuilding, which is still very popular for controlling estrogen. This agent is available both in liquid form and in tablets. Its dosage is usually from 0.25 to 1.0 mg once, with a frequency of one every one / two days.
One tablet with a film coating contains 1 mg of anastrozole. Other ingredients: lactose monohydrate, povidone, sodium starch glycolate, magnesium stearate, hypromellose, macrogol 300, titanium dioxide (E171).
How does it work?
As a result of the use of Anastrozole, estrogen biosynthesis decreases in peripheral tissues and, thus, decreases their plasma concentration, which prevents the development of estrogen-dependent tumors.
The drug is rapidly absorbed from the gastrointestinal tract, reaching a maximum plasma concentration after 2 hours. Plasma protein binding occurs at 40%. The biological half-life is 40-50 hours. Metabolism of the drug occurs in the liver.
After about 7 days of using anastrozole, it reaches a stable plasma concentration. Because of this, you can start using it simultaneously with the launch of SAA. Anastrozole is very dependent on hemoglobin hormones, so doctors use it only in postmenopausal women.
Buy anastrozole (anastrozole for sale)
What do you need to know before you order anastrozole for sale?
When you should not use Anastrozole:
1. If you are allergic to anastrozole or any other ingredient of this drug.
2. Do not use during pregnancy and breastfeeding.
3. It is not recommended to drink alcohol when using drugs.
4. If there is breast cancer, but has not entered menopause.
5. Ischemic heart disease, a condition that can block blood flow to the heart muscle.
6. Osteoporosis or prone to bone fractures.
If any of the above situations apply to you, do not use the drug Anastrozole. If in doubt, consult your doctor or pharmacist before you buy anastrozole.
Arimidex is widely available on prescription and in black markets. In the US, it is not classified as a controlled substance, but you will need a prescription for it to be legally obtained. As for anastrozole buy online or on the black market, almost all anabolic steroid suppliers sell Anastrozole or another brand Arimidex.
Where can i buy anastrozole without a prescription?
In recent years, the ability to buy anastrozole from research chemical laboratories (RCL) has become very popular. RCL produces various uncontrolled substances in a liquid state, often highly concentrated. Anastrozole for sale online legally is only possible for research purposes. This is obviously a loophole in the law that many users of anabolic steroids use.
Where can i buy anastrozole online?
Athletes buy anastrozole online, through anabolic steroid sites or RCL. The connection is rarely faked, so it’s not hard to find a good quality product. However, if you want to buy drug from a steroid supplier - this is not legal. In addition, although the purchase at RCL is in fact legal, only for research purposes, and this can be a problem for the buyer if law enforcement agencies want to check. In any case, the best way to buy the drug will always be through a pharmacy based on the prescription given by your doctor.
H3 Anastrozole dosage
What is the recommended anastrozole dosage? How to safely use this drug? How long to use?
Anastrozole comes in the form of 1 milligram (mg) tablets and is usually taken once a day for medical purposes. It can be taken before, on time or after a meal.
• for men - 0.5 mg - 3 mg;
• for women - 1 mg / day.
Athletes during PCT usually start with a higher dose, and then gradually reduce the dosage. A PCT course usually runs from 7 to 14 days.
In clinical studies, it was noted that daily Anastrozole dosage - 1 mg leads to 80% suppression of estrogen.
The correct dosage of the drug is associated with a gradual increase in dose. The most common practice is 0.25–1 mg every 1–3 days, depending on the purpose of use and the effects observed. At high doses, drug intake should be gradually reduced, as the sudden withdrawal of the agent can lead to an increase in estrogen production that is too rapid. Always use anastrozole as recommended by your doctor.
Anastrozole side effects
Like all drugs of this type, Anastrozole has its drawbacks, despite the fact that it is much better tolerated by the body.
General Anastrozole side effects include:
1. Hot flashes.
3. Pain in the bones and joints, as well as in other areas of the body.
4. Stomach pain, nausea, vomiting or diarrhea.
6. Infection of the throat.
8. Infectious disease.
9. Reduces HDL.
10. Increases weight.
11. Abnormal sensations and tingling in the legs and arms.
12. Swollen lymph nodes.
Serious anastrozole side effects include:
1. The fragility of the bones.
3. Thick blood and chest pain.
4. Stroke, heart attack and high blood pressure.
5. Low red blood cell and white blood cell count.
7. Stevens-Johnson syndrome.
9. Inflammation of the liver.
When using anastrozole, you should avoid taking the following drugs:
1. Supplement DHEA (dihydroepiandrosterone).
2. Soltamox (tamoxifen).
3. Any drugs containing estrogen (birth control pills, drugs for hormone replacement therapy).
4. Warfarin (Coumadin, Jantoven).
Arimidex can slow down the absorption of other drugs, which can lead to an increase in the level of other drugs in the blood.
You should avoid grapefruit and grapefruit juice during taking anastrozole, because together they slow down the body's ability to process certain drugs.
Anastrozole for men
Anastrozole for men is sometimes used to treat breast cancer in men, but has not been well studied in this area. It has been studied for the treatment of male infertility (to balance testosterone levels and maintain a healthy sperm count).
Some male athletes and bodybuilders who use steroids to build muscle and take anastrozole to reduce the production of estrogen, which are a side effect of the use of anabolic steroids.
An increase in estrogen levels causes - a reduction in the testicles, penis, and breast augmentation.
Аnastrozole for men
Anastrozole - is a very convenient agent for men using anabolic steroids, much more effective than Nolvadex or Proviron. Already one dose per day gives excellent results. For some men, even a dose of 0.125 mg per day is enough to overcome the effect of strongly flavoring androgens, Diananbol or testosterone. The use of the drug very effectively blocks water retention and reduces the risk of gynecomastia, and the use of finasteride also brings very good results. One blocks the conversion to estrogen, the second blocks 5-alpha recovery. Together, they effectively minimize the potential side effects of androgens. When using this combination, testosterone will retain its strength. As a result, the resulting muscle mass will be much better without unnecessary water retention.
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